Science

2012

  • . Niphatenones, glycerol ethers from the sponge Niphates digitalis block androgen receptor transcriptional activity in prostate cancer cells: structure elucidation, synthesis, and biological activity. J Med Chem 2012

2011

  • . Small molecule inhibitors targeting the “Achilles’ heel” of androgen receptor activity. ancer Res 2011

2010

  • . Regression of castrate-recurrent prostate cancer by a small molecule inhibitor of the amino-terminus domain of the androgen receptor. Cancer Cell 2010